冬凌草甲素研究进展 |
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引用本文: | 刘淑云,谭英姿,范明松,陈明苍,吴斌.冬凌草甲素研究进展[J].中国当代医药,2012,19(13):17-18,20. |
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作者姓名: | 刘淑云 谭英姿 范明松 陈明苍 吴斌 |
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作者单位: | 1. 上海中医药大学附属曙光医院,上海,201203;中国科学院上海药物研究所,上海,201203 2. 上海中医药大学附属曙光医院,上海,201203 3. 中国科学院上海药物研究所,上海,201203 |
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摘 要: | 冬凌草甲素是从唇形科香茶菜属植物中提取出来的一种对映-贝壳杉烷型二萜类化合物,具有多种药理作用,尤其是抗肿瘤活性。本文对冬凌草甲素的衍生物、药效学及药代动力学等方面进行综述,并对冬凌草甲素的研究开发前景进行展望。
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关 键 词: | 冬凌草甲素 化学结构 药效学 药代动力学 |
Advances in the research of oridonin |
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Authors: | LIU Shuyun TAN Yingzi FAN Mingsong CHEN Mingcang WU Bin |
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Institution: | 1.Shuguang Hospital Affiliated to Shanghai University of Traditional Chinese Medicine,Shanghai 201203,China;2.Shanghai Institute of Materia Medica,Chinese Academy of Sciences,Shanghai 201203,China |
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Abstract: | Oridonin is an ent-kaurene diterpenoid isolated from Rabdosia rubescens (Hemal.) Hara.It has a variety of pharmacological effects,especially its anti-tumor activity.This paper discusses the chemical structure,pharmacodynamics and pharmacokinetics of oridonin.In addition,the development of oridonin in the future is also prospected. |
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Keywords: | Oridonin Chemical structure Pharmacodynamics Pharmacokinetics |
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