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Sorafenib is an inhibitor of UGT1A1 but is metabolized by UGT1A9: implications of genetic variants on pharmacokinetics and hyperbilirubinemia
Authors:Peer Cody J  Sissung Tristan M  Kim Aerang  Jain Lokesh  Woo Sukyung  Gardner Erin R  Kirkland C Tyler  Troutman Sarah M  English Bevin C  Richardson Emily D  Federspiel Joel  Venzon David  Dahut William  Kohn Elise  Kummar Shivaani  Yarchoan Robert  Giaccone Giuseppe  Widemann Brigitte  Figg William D
Affiliation:Clinical Pharmacology Program, Pharmacology and Experimental Therapeutics Section, Molecular Pharmacology Section, Biostatistics and Data Management Branch, Medical Oncology Branch, and HIV/AIDS Malignancy Branch, National Cancer Institute, Bethesda, MD 20892, USA.
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