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Novel bifunctional quinolonyl diketo acid derivatives as HIV-1 integrase inhibitors: design, synthesis, biological activities, and mechanism of action
Authors:Di Santo Roberto  Costi Roberta  Roux Alessandra  Artico Marino  Lavecchia Antonio  Marinelli Luciana  Novellino Ettore  Palmisano Lucia  Andreotti Mauro  Amici Roberta  Galluzzo Clementina Maria  Nencioni Lucia  Palamara Anna Teresa  Pommier Yves  Marchand Christophe
Institution:Istituto Pasteur-Fondazione Cenci Bolognetti, Dipartimento di Studi Farmaceutici, and Istituto di Microbiologia, Università di Roma La Sapienza, P. le A. Moro 5, I-00185 Roma, Italy. roberto.disanto@uniroma1.it
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