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市售DPP-4抑制剂类抗糖尿病药物的比较研究
引用本文:王欣,崔立迁.市售DPP-4抑制剂类抗糖尿病药物的比较研究[J].天津药学,2014(2):75-78.
作者姓名:王欣  崔立迁
作者单位:天津生物工程职业技术学院;天津市产品质量监督检测技术研究院
摘    要:DPP-4抑制剂是近年来上市的一类高效、高选择性抗2型糖尿病药物,通过检索文献,综述已上市的五种DPP-4抑制剂在结构、药代药动、选择性、药物相互作用、副作用等方面的差异.

关 键 词:DPP-4抑制剂  2型糖尿病  西格列汀  沙格列汀  维格列汀  利格列汀  阿格列汀

Comparison of several marketed DPP-4 inhibitors
Wang Xin;Cui Liqian.Comparison of several marketed DPP-4 inhibitors[J].Tianjin Pharmacy,2014(2):75-78.
Authors:Wang Xin;Cui Liqian
Institution:Wang Xin;Cui Liqian;Tianjin Vocational College of Bioengineering;Tianjin Product Quality Inspection Technology Research Institute;
Abstract:DPP - 4 inhibitors, developed in recent years, are a class of anti - diabetes drugs of type 2 diabetes with high effi- ciency and selectivity. By means of summarizing the literatures, differences of five marketed dipeptidyl peptidase - 4 ( DPP - 4 ) inhibitors in structures, dynamic, selectivity, metabolism, and drug- drug interaction were reviewed in this paper.
Keywords:DPP-4 inhibitor  type 2 diabetes  saxagliptin  sitagliptin  linagliptin  vildagliptin  alogliptin
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