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Discovery of INCB3284, a Potent,Selective, and Orally Bioavailable hCCR2 Antagonist
Authors:Chu-Biao Xue  Hao Feng  Ganfeng Cao  Taisheng Huang  Joseph Glenn  Rajan Anand  David Meloni  Ke Zhang  Lingquan Kong  Anlai Wang  Yingxin Zhang  Changsheng Zheng  Michael Xia  Lihua Chen  Hiroyuki Tanaka  Qi Han  D. J. Robinson  Dilip Modi  Lou Storace  Lixin Shao  Vaqar Sharief  Mei Li  Laurine G. Galya  Maryanne Covington  Peggy Scherle  Sharon Diamond  Tom Emm  Swamy Yeleswaram  Nancy Contel  Kris Vaddi  Robert Newton  Greg Hollis  Steven Friedman  Brian Metcalf
Affiliation:Incyte Corporation, Experimental Station E336, Wilmington, Delaware 19880, United States
Abstract:
Keywords:CCR2   chemokine   antagonist   hERG   oral absorption
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