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Allosteric enhancers for A1 adenosine receptor |
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| Authors: | Baraldi Pier Giovanni Iaconinoto Maria Antonietta Moorman Allan R Carrion Maria Dora Cara Carlota Lopez Preti Delia López Olga Cruz Fruttarolo Francesca Tabrizi Mojgan Aghazade Romagnoli Romeo |
| Affiliation: | Dipartimento di Scienze Farmaceutiche, Università di Ferrara, Ferrara, Italy. baraldi@unife.it |
| Abstract: | Allosteric enhancers at the adenosine A(1) receptor have received attention as anti-arrhythmic cardiac agents, and, more recently, as anti-lipolytic agents. In addition, allosteric modulators at the adenosine A(1) receptor have therapeutic potential as analgesics and neuroprotective agents. In particular, the compounds with improved potency as enhancers and reduced antagonist properties are mentioned. |
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| 本文献已被 PubMed 等数据库收录！ | |