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Novel N-Substituted Benzimidazolones as Potent,Selective, CNS-Penetrant,and Orally Active M1 mAChR Agonists |
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| Authors: | Brian Budzik Vincenzo Garzya Dongchuan Shi Graham Walker Marie Woolley-Roberts Joanne Pardoe Adam Lucas Ben Tehan Ralph A. Rivero Christopher J. Langmead Jeannette Watson Zining Wu Ian T. Forbes Jian Jin | |
| Affiliation: | GlaxoSmithKline, 1250 South Collegeville Road, Collegeville, Pennsylvania 19426 | |
| Abstract: | ||
| Keywords: | M1 muscarinic acetylcholine receptor M1 mAChR CNS-penetrant and orally active M1 mAChR agonists subtype selective benzimidazolones 1-(N-substituted piperidin-4-yl)benzimidazolones | |