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Assessing the chemical-induced estrogenicity using in silico and in vitro methods
Institution:1. ProtoQSAR SL., CEEI (Centro Europeo de Empresas Innovadoras), Parque Tecnológico de Valencia, 12 Av. Benjamin Franklin, 46980, Paterna, Valencia, Spain;2. Department of Food Science, Faculty of Veterinary Medicine-FARAH, University of Liège, 10 Av. Cureghem, 4000, Sart-Tilman, Liège, Belgium;3. The Institute for Global Food Security, School of Biological Sciences, Queen''s University Belfast, 19 Chlorine Gardens, BT9 5DL, Belfast, Northern Ireland, United Kingdom;4. MolDrug AI Systems SL, 45 Olimpia Arozena Torres, 46018, Valencia, Spain;1. Graduate School of Global Environmental Studies, Kyoto University, Japan;2. Graduate School of Engineering, Kyoto University, Japan;1. Dep. of Pharmacology and Toxicology, Faculty of Pharmacy, Mansoura University, Mansoura, Egypt;2. Dep. of Pharmacology, Faculty of Pharmacy, Horus University-Egypt, New Damietta, Egypt;1. Department of Computer Sciences, Faculty of Informatics, Camaguey University, Camaguey City, 74650, Camaguey, Cuba;2. Unit of Computer-Aided Molecular “Biosilico” Discovery and Bioinformatic Research (CAMD-BIR Unit), Faculty of Chemistry-Pharmacy. Universidad Central “Martha Abreu” de Las Villas, Santa Clara, 54830, Villa Clara, Cuba;3. Departamento de Química, Universidade Federal de Lavras, CP 3037, 37200-000, Lavras, MG, Brazil;4. Universidad San Francisco de Quito (USFQ), Grupo de Medicina Molecular y Traslacional (MeM&T), Colegio de Ciencias de la Salud (COCSA), Escuela de Medicina, Edificio de Especialidades Médicas, Av. Interoceánica Km 12 ½, Cumbayá, Ecuador;5. Department of Systems and Computer Engineering, Carleton University, Ottawa, Ontario, Canada;6. Unidad de Toxicologia Experimental, Universidad de Ciencias Médicas de Villa Clara Santa Clara, 50200, Villa Clara, Cuba;1. Department of Orthopedics, The Affiliated Wuxi No. 2 People’s Hospital of Nanjing Medical University, Wuxi, 214000, China;2. Department of Neurology, The Affiliated Hospital of Xuzhou Medical University, Xuzhou, Jiangsu, 221000, China;3. Wuxi Center for Disease Control and Prevention, Wuxi, 214000, China;4. Departments of Orthopaedis, The Second Affiliated Hospital of Soochow University, 1055 Sanxiang Road, 2015004, Suzhou, China;5. The Affiliated Wuxi Clinical College of Nantong University, Jiangsu, 214000, China
Abstract:
Keywords:Estrogen receptor  Endocrine disruptor  Persistent organic pollutant  QSAR  Reporter gene assay  Predictive toxicology
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