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Design, synthesis and biological evaluation of heteroaryl diketohexenoic and diketobutanoic acids as HIV-1 integrase inhibitors endowed with antiretroviral activity
Authors:Di Santo R  Costi R  Artico M  Ragno R  Greco G  Novellino E  Marchand C  Pommier Y
Affiliation:Istituto Pasteur-Fondazione Cenci Bolognetti, Dipartimento di Studi Farmaceutici, Università degli Studi di Roma La Sapienza, P.le A. Moro 5, I-00185 Rome, Italy. roberto.disanto@uniroma1.it
Abstract:
Keywords:Integrase inhibitors   Anti-HIV agents   Pyrrole derivatives   Indole derivatives   Diketoacid derivatives
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