转运体和核受体影响药物代谢的研究进展 |
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作者姓名: | 周雪姣 段雅彬 张娟玲 李向阳 |
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作者单位: | 1. 青海大学生态环境工程学院,青海 西宁,810016;2. 青海大学医学院,青海 西宁,810001 |
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基金项目: | 国家自然科学基金项目(81460568),青海省自然科学基金(2016-ZJ-902) |
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摘 要: | 转运体是存在于体内几乎所有器官上的有转运功能的蛋白,对药物在体内的吸收、分布、代谢和排泄有非常重要的作用.而核受体是存在于细胞内的配体依赖性转录因子,可以激活配体影响代谢酶和转运体的表达和活性,进而影响药物在机体内代谢.本文综述了转运体和核受体家族中几个重要的成员以及它们对药物代谢影响的研究进展.
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关 键 词: | 转运体 核受体 药物代谢 |
Progress in the effect of drug metabolism on the transporters and nuclear receptors |
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Authors: | ZHOU Xuejiao DUAN Yabin ZHANG Juanling and LI Xiangyang |
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Institution: | 1. College of Ecological and Environment Engineering, Qinghai University, Xining 810016, China; 2. Medical College of Qinghai University, Xining 810001, China,1. College of Ecological and Environment Engineering, Qinghai University, Xining 810016, China; 2. Medical College of Qinghai University, Xining 810001, China,1. College of Ecological and Environment Engineering, Qinghai University, Xining 810016, China; 2. Medical College of Qinghai University, Xining 810001, China and 1. College of Ecological and Environment Engineering, Qinghai University, Xining 810016, China; 2. Medical College of Qinghai University, Xining 810001, China |
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Abstract: | |
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Keywords: | Transporters Nuclear receptors Drug metabolism |
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