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Biodistribution, toxicity and radiation dosimetry studies of the serotonin transporter radioligand 4-[18F]-ADAM in rats and monkeys
Authors:Ya-Yao Huang  Kuo-Hsing Ma  Ta-Wei Tseng  Ta-Kai Chou  Hanna Ng  Jon C. Mirsalis  Ying-Kai Fu  Tieh-Chi Chu  Wen-Sheng Huang  Chyng-Yann Shiue
Affiliation:(1) PET Center, Department of Nuclear Medicine, Tri-Service General Hospital, 325 Sec. 2, Cheng-Kung Rd., Neihu 114, Taipei, Taiwan;(2) Department of Biomedical Engineering and Environmental Sciences, National Tsing Hua University, 101 Sec. 2, Kuang-Fu Rd., Hsinchu, 30013, Taiwan;(3) Department of Biology and Anatomy, National Defense Medical Center, Taipei, Taiwan;(4) SRI International, 333 Ravenswood Avenue, Menlo Park, CA 94025, USA;(5) Institute of Nuclear Energy Research, 1000, Wenhua Rd., Taoyuan, 32546, Taiwan;(6) Department of Chemistry, Chung Yuan Christian University, Chung-Li, Taiwan;(7) Department of Radiological Technology, Yuanpei University, 306, Yuanpei St., Hsinchu, Taiwan;(8) Department of Radiology, University of Pennsylvania, 3400 Spruce St., Philadelphia, PA 19104, USA
Abstract:

Purpose  

4-[18F]-ADAM is a potent serotonin transport imaging agent. We studied its toxicity in rats and radiation dosimetry in monkeys before human studies are undertaken.
Keywords:
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