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Discovery of a subtype-selective,covalent inhibitor against palmitoylation pocket of TEAD3
Authors:Tian Lu  Yong Li  Wenchao Lu  TWGM Spitters  Xueyu Fang  Jun Wang  Simian Cai  Jing Gao  Yanting Zhou  Zhe Duan  Huan Xiong  Liping Liu  Qi Li  Hualiang Jiang  Kaixian Chen  Hu Zhou  Hua Lin  Huijin Feng  Bing Zhou  Christopher L Antos  Cheng Luo
Institution:1. School of Chinese Materia Medica, Nanjing University of Chinese Medicine, Nanjing 210023, China;2. The Center for Chemical Biology, Drug Discovery and Design Center, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China;3. Department of Medicinal Chemistry, State Key Laboratory of Drug Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China;4. Department of Cancer Biology, Dana-Farber Cancer Institute, Boston, MA 02215, USA;5. School of Life Science and Technology, ShanghaiTech University, Shanghai 201210, China;6. School of Life Sciences and Biotechnology, Shanghai Jiao Tong University, Shanghai 200240, China;7. Department of Analytical Chemistry and CAS Key Laboratory of Receptor Research, Shanghai Institute of Materia Medica, Chinese Academy of Sciences, Shanghai 201203, China;8. School of Pharmacy, Nanchang University, Nanchang 330006, China;9. Pharmacological and Toxicological Chemistry and Biochemistry Laboratory, UMR 8601 CNRS, University of Paris, Paris Cedex 06, 75270, France;10. School of Pharmaceutical Science and Technology, Hangzhou Institute for Advanced Study, University of Chinese Academy of Sciences, Hangzhou 310024, China
Abstract:
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