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Molecular mechanism by which the K70E mutation in human immunodeficiency virus type 1 reverse transcriptase confers resistance to nucleoside reverse transcriptase inhibitors 下载免费PDF全文
Sluis-Cremer N Sheen CW Zelina S Torres PS Parikh UM Mellors JW 《Antimicrobial agents and chemotherapy》2007,51(1):48-53
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Stampidine is a potent inhibitor of Zidovudine- and nucleoside analog reverse transcriptase inhibitor-resistant primary clinical human immunodeficiency virus type 1 isolates with thymidine analog mutations 总被引:2,自引:0,他引:2 下载免费PDF全文
Uckun FM Pendergrass S Venkatachalam TK Qazi S Richman D 《Antimicrobial agents and chemotherapy》2002,46(11):3613-3616
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Molecular mechanisms of tenofovir resistance conferred by human immunodeficiency virus type 1 reverse transcriptase containing a diserine insertion after residue 69 and multiple thymidine analog-associated mutations 总被引:3,自引:0,他引:3 下载免费PDF全文
White KL Chen JM Margot NA Wrin T Petropoulos CJ Naeger LK Swaminathan S Miller MD 《Antimicrobial agents and chemotherapy》2004,48(3):992-1003
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Gln145Met/Leu changes in human immunodeficiency virus type 1 reverse transcriptase confer resistance to nucleoside and nonnucleoside analogs and impair virus replication 下载免费PDF全文
Paolucci S Baldanti F Maga G Cancio R Zazzi M Zavattoni M Chiesa A Spadari S Gerna G 《Antimicrobial agents and chemotherapy》2004,48(12):4611-4617
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Effects of specific zidovudine resistance mutations and substrate structure on nucleotide-dependent primer unblocking by human immunodeficiency virus type 1 reverse transcriptase 下载免费PDF全文
Meyer PR Matsuura SE Tolun AA Pfeifer I So AG Mellors JW Scott WA 《Antimicrobial agents and chemotherapy》2002,46(5):1540-1545
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Sequence diversity of the reverse transcriptase of human immunodeficiency virus type 1 from untreated Brazilian individuals. 下载免费PDF全文
Rodrigo Brindeiro Bart Vanderborght Elena Caride Letícia Correa Rejane M. Oravec Oscar Berro Lieven Stuyver Amilcar Tanuri 《Antimicrobial agents and chemotherapy》1999,43(7):1674-1680
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Selective interaction of the human immunodeficiency virus type 1 reverse transcriptase nonnucleoside inhibitor efavirenz and its thio-substituted analog with different enzyme-substrate complexes 下载免费PDF全文
Maga G Ubiali D Salvetti R Pregnolato M Spadari S 《Antimicrobial agents and chemotherapy》2000,44(5):1186-1194
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Variations in reverse transcriptase and RNase H domain mutations in human immunodeficiency virus type 1 clinical isolates are associated with divergent phenotypic resistance to zidovudine 下载免费PDF全文
Ntemgwa M Wainberg MA Oliveira M Moisi D Lalonde R Micheli V Brenner BG 《Antimicrobial agents and chemotherapy》2007,51(11):3861-3869
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TMC125, a novel next-generation nonnucleoside reverse transcriptase inhibitor active against nonnucleoside reverse transcriptase inhibitor-resistant human immunodeficiency virus type 1 下载免费PDF全文
Andries K Azijn H Thielemans T Ludovici D Kukla M Heeres J Janssen P De Corte B Vingerhoets J Pauwels R de Béthune MP 《Antimicrobial agents and chemotherapy》2004,48(12):4680-4686