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High specific activity tritium labeling of anti‐tumor agent CEP‐2563 |
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| Abstract: | [Ester Methylene‐3H] CEP‐2563 ( 9 ) was synthesized by the tritiation of precursor 6 with NaB3H4 followed by esterification with BOC‐Lys(BOC)‐β‐Ala‐OH and deprotection. Copyright © 2005 John Wiley & Sons, Ltd. |
| Keywords: | anti‐tumor CEP‐751 CEP‐2563 NaB3H4 tritium |