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Etravirine inhibits ABCG2 drug transporter and affects transplacental passage of tenofovir disoproxil fumarate
Institution:1. Endacea Inc., 2 Davis Drive, P.O. Box 12076, Research Triangle Park, NC 27709-2076, United States;2. Department of Medicine Brigham and Women?s Hospital 75 Francis Street, Boston MA 02115, United States;3. Saint Louis University School of Medicine, St. Louis MO, United States;1. Dana Farber Cancer Institute and Harvard Medical School, Boston, MA, USA;2. Comprehensive Cancer Center, University of Alabama at Birmingham, Birmingham, AL, USA;1. Division of Cardiovascular Surgery, Shiga University of Medical Science, Setatsukinowa, Otsu, Japan;2. Department of Pharmacology, Shiga University of Medical Science, Setatsukinowa, Otsu, Japan;3. Department of Anatomy, Shiga University of Medical Science, Setatsukinowa, Otsu, Japan;1. Department of Pharmacological and Pharmaceutical Sciences, College of Pharmacy, University of Houston, Houston, TX 77030, USA;2. Pfizer, Groton, CT 06340, USA;1. Department of Clinical Pharmacology, College of Pharmacy, Dalian Medical University, China;2. Provincial Key Laboratory for Pharmacokinetics and Transport, Liaoning, Dalian Medical University, China;3. Research Institute of Integrated Traditional and Western Medicine of Dalian Medical University, Liaoning, China;1. Magee-Womens Research Institute, University of Pittsburgh, Pittsburgh, PA, USA;2. Department of Obstetrics, Gynecology and Reproductive Sciences, University of Pittsburgh, Pittsburgh, PA, USA;3. Department of Microbiology and Molecular Genetics, University of Pittsburgh, Pittsburgh, PA, USA
Abstract:
Keywords:P-glycoprotein  Breast cancer resistance protein  Pregnancy  Tenofovir disoproxil fumarate  Abacavir  Transplacental pharmacokinetics
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